Publication List
Original Papers
1. Takayuki Doi, Masahito Yoshida, Ichiro Hijikuro, and Takashi Takahashi:
An Efficient Synthesis of Polymer-Supported Silyl Linkers Using
a Di-Grignard Reagent,
Tetrahedron Lett., 45 (29), 5723-5726 (2004).
2. Takayuki Doi, Masahito Yoshida, Ichiro Hijikuro, and Takashi Takahashi:
Selective
Capture of 1α, 25-(OH)2-Previtamin D3 Utilizing Polymer-Supported Trialkylsilyl Triflate in the Synthesis of 1α, 25-(OH)2-Vitamin D3,
Tetrahedron Lett., 45 (29), 5727-5729 (2004).
3. Takayuki Doi, Masahito Yoshida, Kazuo
Shin-ya, and Takashi Takahashi:
Total Synthesis of (R)-Telomestatin,
Org. Lett., 8 (18), 4165-4167 (2006). (Highlighted in ChemInform
issue 38/04)
4. Masahito Yoshida, Takayuki Doi, Sungmin
Kang, Junji Watanabe, and Takashi Takahashi:
Solid-Phase Combinatorial Synthesis of Ester-Type Banana-Shaped
Molecule by Way of Sequential Palladium-Catalyzed Carbonylation,
Chem. Commun., 2756-2758
(2009).
5. Masahito Yoshida, Christian Hedberg, Markus Kaiser, and
Herbert Waldmann:
Traceless Solid-Phase Synthesis on Natural Product Inspired
cis-1,2-Dehydrodecalines,
Chem. Commun., 2926-2928
(2009). (Highlighted in Synfacts issue 2009/08)
6. Kazuaki Shibata, Masahito Yoshida,
Takayuki Doi, and Takashi Takahashi:
Derivatization of a Tris-Oxazole Using Pd-catalyzed Coupling
Reactions of a 5-Bromooxazole Moiety,
Tetrahedron Lett., 51 (13), 1674-1677 (2010). (Highlighted in ChemInform
issue 41/29)
7. Masahito Yoshida, Hisayuki
Ishida, Yoshitaka Ishida, Yoko Yashiroda, Minoru
Yoshida, Motoki Takagi, Kazuo Shin-ya, and Takayuki
Doi:
Synthesis, Structure Determination and Biological Evaluation of Destruxin E,
Org. Lett., 12 (17), 3792-3795 (2010).
8. Shin-ichiro Fuse, Nobutake Tanabe, Masahito Yoshida, Hayato Yoshida, Takayuki Doi, and Takashi Takahashi:
Continuous-Flow Synthesis of Vitamin D3,
Chem. Commun., 46 (46),
8722-8724 (2010).
9. Takayuki Doi, Kazuaki Shibata, Masahito
Yoshida, Motoki Takagi, Masayuki Tera, Kazuo Nagasawa, Kazuo Shin-ya, and Takashi Takahashi:
(S)-Stereoisomer of Telomestatin
as a Potent G-quadrulex Binder and Telomerase
Inhibitor,
Org. Biomol. Chem., 9
(2), 387-393 (2011).
10. Ikuko Kozone, Miho Izumikawa, Keiichiro Motohashi,
Aya Nagai, Masahito Yoshida, Takayuki Doi, Motoki Takagi, and Kazuo Shin-ya:
Isolation of New Hexapeptides-JBIR-39 and 40- from a Marine
Sponge-Derived Streptomyces sp. Sp080513SC-24,
J. Marine Sci. Res. Development, 1:101. doi: 10.4172/2155-9910.1000101 (2011).
11. Masahito Yoshida, Yuta Fujino,
and Takayuki Doi:
Synthesis of g-Benzopyranone by TfOH-promoted
Regioselective Cyclization of o-Alkynoylphenols,
Org. Lett., 13 (17), 4526-4529 (2011). (Highlighted in ChemInform
issue 43/01)
12. Masahito Yoshida, Yuta Fujino,
Koya Saito, and Takayuki Doi:
Regioselective Synthesis of Flavone Derivatives via
DMAP-catalyzed Cyclization of o-Alkynoylphenols,
Tetrahedron, 67 (51), 9993-9997 (2011). (Highlighted in ChemInform
issue 43/17)
13. Takayuki Doi, Terushige Muraoka, Taichi Oshiro, Daisuke Matsuda, Masahito Yoshida,
Takashi Takahashi, Satoshi Omura, and Hiroshi Tomoda:
Conformationally Restricted Analog and Biotin-Labeled Probe
Based on Beauveriolide III,
Bioorg.
Med. Chem. Lett., 22 (1), 696-699 (2012).
14. Takayuki Doi, Kouya Oikawa,
Jun Suzuki, Masahito Yoshida, and Nobuhiko Iki:
Development of a Near Infrared Fluorescence Labelling Reagent:
Synthesis of Indole-Functionalized Indocyanine Green Derivatives,
Synlett,
(2), 306-310 (2012).
15. Masahito Yoshida, Koya Saito,
Yuta Fujino, and Takayuki Doi:
A Concise Synthesis of 3-Aroylflavone via Lewis Base
9-Azajulolidine-catalyzed Tandem Acyl Transfer-Cyclization,
Chem. Commun., 48 (96),
11796-11798 (2012). (Highlighted
in ChemInform issue 44/14)
16. Kosuke Ohsawa, Masahito Yoshida,
and Takayuki Doi:
A Direct and Mild Formylation Method for Substituted Benzenes
Utilizing Dichloromethyl Methyl Ether-Silver Trifluoromethanesulfonate,
J. Org. Chem., 78 (7), 3438-3444 (2013). (Highlighted in ChemInform
issue 44/32)
17. Kazuaki Shibata, Masahito Yoshida, Takashi Takahashi, Motoki
Takagi, Kazuo Shin-ya, and Takayuki Doi:
Synthesis of Hepta-Oxazole Macrocyclic Analogues of Telomestatin and Evaluation of Their Telomerase Inhibitory
Activities,
Bull. Chem. Soc. Jpn., 86
(12), 1453-1465 (2013).
18. Masahito Yoshida, Hiroshi Sato, Yoshitaka Ishida,
Hiroshi Nakagawa, and Takayuki Doi:
Scalable Solution-Phase Synthesis of Biologically Active Cyclodepsipeptide Destruxin E, a
Potent Negative Regulator of Osteoclast Morphology,
J. Org. Chem., 79 (1), 296-306 (2014).
19. Takayuki Doi, Masahito Yoshida, Kosuke Ohsawa,
Kazuo Shin-ya, Motoki Takagi, Yoshinori Uekusa, Takumi Yamaguchi, Koichi Kato, Takatsugu
Hirokawa, and Tohru Natsume:
Total Synthesis and Characterization of Thielocin
B1 as a Protein-Protein Interaction Inhibitor of PAC3 Homodimer,
Chem. Sci., 5 (5), 1860-1868 (2014).
20. Mokoto Kobayashi, Masato Nishizawa, Nao Inoue,
Takahiro Hosoya, Masahito Yoshida, Yuko Sagesaka, Takayuki Doi, Tsutomu Nakayama, Shigenori Kumazawa, and Ikuo Ikeda:
Epigallocatechin Gallate Decreases the Micellar Solubility of
Cholesterol via Specific Interaction with Phosphatidylcholine,
J. Agric. Food Chem., 62 (13), 2881-2890 (2014).
21. Masahito Yoshida, Koya Saito,
Yuta Fujino, and Takayuki Doi:
A Concise Total Synthesis of Biologically Active Frutinones via Tributylphosphine-catalyzed
Tandem Acyl Transfer-Cyclization,
Tetrahedron, 70 (21), 3452-3458 (2014). (Highlighted in ChemInform
issue 45/43)
22. Masahito Yoshida, Hiroyuki Otaka,
and Takayuki Doi:
An Efficient Partial Reduction of a, b-Unsaturated Esters Using DIBAL-H in Flow,
Eur. J. Org. Chem., (27), 6010-6016 (2014). (Highlighted in ChemInform
issue 46/12)
23. Yuichi Masuda, Jun Suzuki, Yuichi Onda,
Yuta Fujino, Masahito Yoshida, and Takayuki
Doi:
Total Synthesis and Conformational Analysis of Apratoxin C,
J. Org. Chem., 79 (17), 7844-7853 (2014).
24. Takayuki Doi, Naoko Yamaguchi, Kosuke Ohsawa,
Kazuoki Nakai, Masahito
Yoshida, Kazuhiro Satake, Yuji Mitani, Hiroshi Nakagawa, Takashi Takahashi, and Toshihisa Ishikawa:
Synthesis and Biological Evaluation of C-Aromataxane
Derivatives as P-Glycoprotein-Mediated Multi Drug Resistance Reversal Agents,
Heterocycles, 90 (1), 482-501 (2015).
25. Koya Saito, Masahito Yoshida, and Takayuki
Doi:
An Efficient Synthesis of Aurone Derivatives by Tributylphosphine-catalyzed Cyclization of o-Alkynoylphenols,
Chem Lett., 44 (2), 141-143 (2015). (Highlighted in ChemInform
issue 46/33)
26. Masahito Yoshida, Naoki Sekioka,
Miho Izumikawa, Ikuko Kozone, Motoki Takagi, Kazuo Shin-ya,
and Takayuki Doi:
Total Synthesis and Structure Elucidation of JBIR-39: A Linear
Hexapeptide Possessing Piperazic Acid and g-Hydroxypiperazic
Acid Residues,
Chem. Eur. J., 21 (7), 3031-3041 (2015).
27. Takayuki Doi, Hiroyuki Otaka, Koji Umeda,
and Masahito Yoshida:
Study for Diastereoselective Aldol Reaction in Flow: Synthesis
of (E)-(S)-3-Hydroxy-7-Tritylthio-4-Heptanoic Acid,
Tetrahedron, 71 (37), 6463-6470 (2015).
28. Masahito Yoshida, Ken-ichi Sasahara, and Takayuki Doi:
Total Synthesis of Cyclodepsipeptide Spiruchostatin A on Silyl-Linked Polymer-Support,
Tetrahedron, 71 (40), 7647-7653 (2015). (Highlighted in Synfacts
issue 2015/12)
29. Masahito Yoshida, Yoshitaka Ishida, Kenta Adachi, Hayato Murase, Hiroshi Nakagawa,
and Takayuki Doi:
Solid-Phase Combinatorial Synthesis and Biological Evaluation of
Destruxin E,
Chem. Eur. J., 21 (50), 18417-18430 (2015).
30. Miho Izumikawa, Teppei
Kawahara, Noritaka Kagaya,
Hideki Yamamura, Masayuki Hayakawa, Motoki Takagi, Masahito Yoshida,
Takayuki Doi, and Kazuo Shin-ya:
Pyrrolidine-Containing Peptides, JBIR-126, -148, and -149 from
Streptomyces sp. NBRC 111228,
Tetrahedron Lett., 56 (39), 5333-5336 (2015). (Highlighted in ChemInform
issue 47/03)
31. Masahito Yoshida, Yuichi Onda,
Yuichi Masuda, and Takayuki Doi:
Potent Oxazoline Analogue of Apratoxin C: Synthesis, Biological Evaluation, and
Conformational Analysis,
Biopolymers-Peptide Science, 106 (4), 404-414
(2016).
32. Yuichi Masuda, Kazumasa Aoyama, Masahito Yoshida, Keisuke
Kobayashi, Taichi Oshiro, Hiroshi Tomoda,
and Takayuki Doi:
Design, Synthesis, and Biological Evaluation of Beauverilide Analogues Bearing Photoactive Amino Acids,
Chem. Pharm. Bull., 64 (7), 754-765 (2016).
33. Hiroshi Sato, Masahito Yoshida, Hayato
Murase, Hiroshi Nakagawa, and Takayuki Doi:
Combinatorial Synthesis and Biological Evaluation of Cyclodepsipeptide Destruxin B as
a Negative Regulator for Osteoclast Morphology,
ACS Combi. Sci., 18 (9), 590-595 (2016).
34. Yuichi Onda, Yuichi Masuda, Masahito
Yoshida, and Takayuki Doi:
Comformational
Design and Synthesis of Apratoxin A
Mimetics Modified at the a, b-Unsaturated Thiazoline
Moiety,
J.
Med. Chem., 60 (15), 6751-6765 (2017).
35. Reiya Taniguchi, Asuka
Inoue, Misa Sayama, Akiharu
Uwamizu, Kunio Hirata, Keitaro
Yamashita, Masahito Yoshida, Yoshiki Tanaka,
Hideaki E. Kato, Yoshiko Nakada-Nakura, Yuko Otani,
Tomohiro Nishizawa, Takayuki Doi, Tomohiko Ohwada,
Ryuichiro Ishitani, Junken
Aoki, and Osamu Nureki:
Structure Insights into Ligand Recognition by the
Lysophosphatidic Acid Receptor LPA6,
Nature, 548 (7667), 356-360 (2017).
36. Masahito Yoshida, Koji Umeda, and Takayuki Doi:
Stereoselective Synthesis of β-Amino Acid Derivatives by
Asymmetric Mannich Reaction in Flow,
Bull. Chem. Soc. Jpn., 90
(10), 1157-1163 (2017).
37. Koya Saito, Masahito Yoshida, Hidehiro Uekusa, and Takayuki
Doi:
Facile Synthesis of Pyrollyl
4-Quinolinone Alkaloids Quinolactacide by
9-AJ-Catalyzed Tandem Acyl Transfer-Cyclization of o-Alkynoylaniline
Derivatives,
ACS Omega, 2 (8), 4370-4381 (2017).
38. Shinya Ito, Koji Ogawa, Koh Takeuchi Motoki Takagi, Masahito
Yoshida, Takatsugu Hirokawa, Shoshiro
Hirayama, Kazuo Shin-ya, Ichiro Shimada, Takayuki
Doi, Naoki Goshima, and Tohru
Natsume:
A Small Compound Inhibiting Collagen-Specific Molecular
Chaperone as a Potential Remedy for Fibrosis,
J. Biol. Chem., 292 (49), 20076-20085 (2017).
39. Masahito Yoshida, Koya Saito, Hikaru Kato, Sachiko Tsukamoto, and Takayuki Doi:
Total Synthesis and Biological Evaluation of Siladenoserinol
A and its Analogues,
Angew.
Chem. Int. Ed., 57 (18), 5137-5140 (2018). (Highlighted in Synfacts issue
2018/06)
40. Kosuke
Ohsawa, Masahito Yoshida, Miho Izumikawa, Motoki Takagi, Kazuo Shin-ya,
Naoki Goshima, Takatsugu
Hirokawa, Tohru Natsume,
and Takayuki Doi:
Synthesis and Biological Evaluation of Thielocin
B1 Analogues as Protein-Protein Interaction Inhibitors of PAC3 Homodimer,
Bioorg.
Med. Chem., 26 (23-24), 6023-6034 (2018).
41. Masahito
Yoshida, Kenta Adachi, Hayato Murase,
Hiroshi Nakagawa, and Takayuki Doi:
Parallel Synthesis and Biological Evaluation of Destruxin E Analogs Modified with a Side Chain in the a-Hydroxycarboxylic Acid Moiety,
Eur. J. Org. Chem., 1669-1676 (2019).
42. Takayuki
Ohyoshi, Keisuke Mitsugi, Tatsuya Higuma,
Fumitaka Ichimura, Masahito Yoshida, and Hideo
Kigoshi:
Concise Total Synthesis of Phelligridin
A, C, and D,
RSC Advances, 9 (18), 7321-7323 (2019).
43. Kosuke
Ohsawa, Masato Sugai, Linnan Zhang, Yuichi Masuda, Masahito Yoshida, and
Takayuki Doi:
Total Synthesis and Structural Revision of Cyclotetrapeptide
Asperterrestide A,
J. Org. Chem., 84 (11), 6765-6779 (2019).
44. Shinya
Ito, Masazumi Saito, Masahito Yoshida, Koh
Takeuchi, Takayuki Doi, and Kazuhiro Nagata:
A BRET-based Assay Reveals Collagen-Hsp47 Interaction Dynamics
in the Endoplasmic Reticulum and Small-Molecule Inhibition of This Interaction,
J.
Biol. Chem., 294 (44), 15962-15972 (2019).
45 Masahito Yoshida:
Combinatorial Synthesis and Biological Evaluation of Destruxins,
Chem.
Pharm. Bull., 67 (10), 1023-1029 (2019).
46 Yuichi Onda, Kazuki Fukushi,
Kosuke Ohsawa, Masahito Yoshida, Yuichi
Masuda, and Takayuki Doi:
Synthesis of A Biphenylalanine
Analogue of Apratoxin A
Displaying Substantially Enhanced Cytotoxicity,
Heterocycles, 101 (2), 679-691 (2020).
47 Masahito Yoshida, Masazumi
Saito, Shinya Ito, Koji Ogawa, Naoki Goshima,
Kazuhiro Nagata, and Takayuki Doi:
Structure-Activity Relationship Study on Col-003, a
Protein-Protein Interaction Inhibitor between Collagen and Hsp47
Chem. Pharm.
Bull., 68 (3), 220-226 (2020).
48 Takayuki
Ohyoshi, Keisuke Mitsugi, Fumitaka Ichimura, Tatsuya Higuma, Masahito
Yoshida, and Hideo Kigoshi:
Total Synthesis and Structure-Activity Relationship Studies of Phelligridin C and D, and Phellifuropyranone
A
Bull. Chem. Soc.
Jpn., 93
(12), 1540-1551
(2020).
(December 2020)